TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 0.00794nMAssay Description:Ability to displace [3H]QNB from HM1 receptor binding to acetylcholine was evaluated by ligand inhibition assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 0.00800nMAssay Description:Ability to displace [3H]QNB from HM1 receptor binding to acetylcholine was evaluated by ligand inhibition assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 0.0129nMAssay Description:Ability to displace [3H]QNB from HM1 receptor binding to acetylcholine was evaluated by ligand inhibition assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 0.0130nMAssay Description:Ability to displace [3H]QNB from HM1 receptor binding to acetylcholine was evaluated by ligand inhibition assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 0.0759nMAssay Description:Ability to displace [3H]QNB from HM1 receptor binding to acetylcholine was evaluated by ligand inhibition assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 0.0760nMAssay Description:Ability to displace [3H]QNB from HM2 receptor binding to acetylcholine was evaluated by ligand inhibition assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 0.229nMAssay Description:Ability to displace [3H]QNB from HM2 receptor binding to acetylcholine was evaluated by ligand inhibition assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 0.229nMAssay Description:Binding of [3H]-QNB to HM2 receptor was evaluated by saturation binding assayMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity against nicotinic acetylcholine receptor (nAChR)Checked by AuthorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 562nMAssay Description:Ability to displace [3H]QNB from HM1 receptor binding to acetylcholine was evaluated by ligand inhibition assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 851nMAssay Description:Ability to displace [3H]QNB from HM2 receptor binding to acetylcholine was evaluated by ligand inhibition assayMore data for this Ligand-Target Pair
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 2.80E+4nMAssay Description:Binding affinity against nicotinic acetylcholine receptor (nAChR)Checked by AuthorMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 6.00E+4nMAssay Description:Inhibition of high affinity dopamine uptake at concentration of 1 microMMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 9.00E+4nMAssay Description:Inhibition constant of high-affinity choline uptakeMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent creatine transporter 1(Rattus norvegicus)
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 1.30E+5nMAssay Description:Inhibition constant of high-affinity 5-HT uptakeMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 3.90E+5nMAssay Description:Inhibition constant of high-affinity 5-HT uptakeMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University of Toledo
Curated by ChEMBL
University of Toledo
Curated by ChEMBL
Affinity DataKi: 5.30E+5nMAssay Description:Inhibition constant of high-affinity dopamine uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+7nMAssay Description:Enzyme inhibition dissociation constant for choline acetyl transferase (ChAcT) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+7nMAssay Description:Enzyme inhibition dissociation constant for choline acetyl transferase (ChAcT) was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of EGFR1 (unknown origin) after 1 hr in presence of adenosine 5'[gamma-33P]triphosphate by microbeta microplate counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of binding of [3H]l-quinuclidinyl benzilate ([3H]L-QNB) to muscarinic acetylcholine receptor of Primary olfactory cortex region of forebra...More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of binding of [3H]L-quinuclidinyl benzilate ([3H]-l-QNB) to muscarinic acetylcholine receptor of dentate gyrus region of forebrainMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of binding of [3H]L-quinuclidinyl benzilate ([3H]-l-QNB) to muscarinic acetylcholine receptor of ventral dentate gyrus region of forebrainMore data for this Ligand-Target Pair